NESS-040C5
NESS-040C5 is a potent cannabinoid agonist which was developed for the treatment of glaucoma.[1] It has reasonable selectivity for the CB2 receptor subtype, having a CB2 affinity of 0.4nM, and 25x selectivity over the related CB1 receptor.[2]
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| Formula | C27H33N3OS |
| Molar mass | 447.64 g·mol−1 |
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See also
References
- Paolo Lazzari et al. Pharmaceutical Compounds. US Patent 8106218
- Hanus LO, Mechoulam R (2010). "Novel natural and synthetic ligands of the endocannabinoid system". Current Medicinal Chemistry. 17 (14): 1341–59. doi:10.2174/092986710790980096. PMID 20166928.
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