Enilospirone
Enilospirone (CERM-3,726) is a selective 5-HT1A receptor agonist of the azapirone class.[1]
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| Routes of administration | Oral |
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| ECHA InfoCard | 100.056.284  |
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| Formula | C15H18ClNO3 |
| Molar mass | 295.76 g·mol−1 |
See also
References
- Maurel JL, Autin JM, Funes P, Newman-Tancredi A, Colpaert F, Vacher B (October 2007). "High-efficacy 5-HT1A agonists for antidepressant treatment: a renewed opportunity". Journal of Medicinal Chemistry. 50 (20): 5024–33. doi:10.1021/jm070714l. PMID 17803293.
Further reading
- Nicholson AN, Stone BM (1982). "6-(3-chloro)-phenoxy-2-methyl-1-oxa-4-azospiro-[4,5]decane-3-one (CERM 3726) and sleep of healthy men". Psychopharmacology. 76 (2): 157–9. doi:10.1007/BF00435270. PMID 6805026. S2CID 666391.
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| GABAAR PAMs |
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| Gabapentinoids (α2δ VDCC blockers) | |
| Antidepressants |
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| Sympatholytics (Antiadrenergics) |
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| Phenylpiperazines |
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| Diphenylalkylpiperazines (benzhydrylalkylpiperazines) |
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| Pyrimidinylpiperazines | |
| Pyridinylpiperazines | |
| Benzo(iso)thiazolylpiperazines | |
| Tricyclics (piperazine attached via side chain) |
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